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Jinfang Tang,Jinhua Zhu 경남대학교 수학교육과 2020 Nonlinear Functional Analysis and Applications Vol.25 No.3
In this paper, a new modified proximal point algorithm involving a finite family of minimization problem and fixed point for a finite family of demicontractive in Hadamard spaces is proposed. Some ∆-convergence and strong convergence theorems for the sequence generated by the algorithm are proved in Hadamard space withr suitable conditions. The results presented in the paper improve and generalize some recent results.
Dong, Wei-Wei,Zhao, Jinhua,Zhong, Fei-Liang,Zhu, Wen-Jing,Jiang, Jun,Wu, Songquan,Yang, Deok-Chun,Li, Donghao,Quan, Lin-Hu The Korean Society of Ginseng 2017 Journal of Ginseng Research Vol.41 No.4
Background: In general, after Panax ginseng is administered orally, intestinal microbes play a crucial role in its degradation and metabolization process. Studies on the metabolism of P. ginseng by microflora are important for obtaining a better understanding of their biological effects. Methods: In vitro biotransformation of P. ginseng extract by rat intestinal microflora was investigated at $37^{\circ}C$ for 24 h, and the simultaneous determination of the metabolites and metabolic profile of P. ginseng saponins by rat intestinal microflora was achieved using LC-MS/MS. Results: A total of seven ginsenosides were detected in the P. ginseng extract, including ginsenosides Rg1, Re, Rf, Rb1, Rc, Rb2, and Rd. In the transformed P. ginseng samples, considerable amounts of deglycosylated metabolite compound K and Rh1 were detected. In addition, minimal amounts of deglycosylated metabolites (ginsenosides Rg2, F1, F2, Rg3, and protopanaxatriol-type ginsenosides) and untransformed ginsenosides Re, Rg1, and Rd were detected at 24 h. The results indicated that the primary metabolites are compound K and Rh1, and the protopanaxadiol-type ginsenosides were more easily metabolized than protopanaxatriol-type ginsenosides. Conclusion: This is the first report of the identification and quantification of the metabolism and metabolic profile of P. ginseng extract in rat intestinal microflora using LC-MS/MS. The current study provided new insights for studying the metabolism and active metabolites of P. ginseng.
Biotransformation of Panax ginseng extract by rat intestinal microflora
Wei-Wei Dong,Jinhua Zhao,Fei-Liang Zhong,Wen-Jing Zhu,Jun Jiang,Songquan Wu,Deok-Chun Yang,Donghao Li,Lin-Hu Quan 고려인삼학회 2017 Journal of Ginseng Research Vol.41 No.4
Background: In general, after Panax ginseng is administered orally, intestinal microbes play a crucial role in its degradation and metabolization process. Studies on the metabolism of P. ginseng by microflora are important for obtaining a better understanding of their biological effects. Methods: In vitro biotransformation of P. ginseng extract by rat intestinal microflora was investigated at 37C for 24 h, and the simultaneous determination of the metabolites and metabolic profile of P. ginseng saponins by rat intestinal microflora was achieved using LCeMS/MS. Results: A total of seven ginsenosides were detected in the P. ginseng extract, including ginsenosides Rg1, Re, Rf, Rb1, Rc, Rb2, and Rd. In the transformed P. ginseng samples, considerable amounts of deglycosylated metabolite compound K and Rh1 were detected. In addition, minimal amounts of deglycosylated metabolites (ginsenosides Rg2, F1, F2, Rg3, and protopanaxatriol-type ginsenosides) and untransformed ginsenosides Re, Rg1, and Rd were detected at 24 h. The results indicated that the primary metabolites are compound K and Rh1, and the protopanaxadiol-type ginsenosides were more easily metabolized than protopanaxatriol-type ginsenosides. Conclusion: This is the first report of the identification and quantification of the metabolism and metabolic profile of P. ginseng extract in rat intestinal microflora using LCeMS/MS. The current study provided new insights for studying the metabolism and active metabolites of P. ginseng.
Lan Zhou,Fuxi Jiang,Jinhua She,Zhu Zhang 제어·로봇·시스템학회 2020 International Journal of Control, Automation, and Vol.18 No.8
This paper presents a generalized-extended-state-observer (GESO)-based repetitive control (RC) method for a direct-current motor servo system (DCMSS) subject to parameter perturbation and load torque variation, which are mismatched. A GESO is constructed to estimate the lumped disturbance in real time fashion. Incorporating the estimate into a state-feedback RC law yields a composite controller with a dynamical compensation gain, which ensures that the suppression of the mismatched total disturbance and the tracking of periodic signal are achieved simultaneously. The stability criterion and design procedure of the system are developed. Finally, simulation results show that the GESO-RC based DCMSS effectively eliminates the influences on the output of the parameter variation and the load disturbance and has both satisfactory dynamical performance and robustness. Comparisons with conventional PID control, PID-RC, and standard extended-state-observer based RC demonstrate the superiority of this method.
Generalized-extended-state-observer-based Sliding-mode Control for Buck Converter Systems
Lan Zhou,Xiaojun Yi,Zhuang Jiang,Zhu Zhang,Jinhua She 제어·로봇·시스템학회 2022 International Journal of Control, Automation, and Vol.20 No.12
This paper presents a generalized-extended-state-observer (GESO)-based sliding-mode control (SMC) method to deal with mismatched parameter uncertainty and reference-input mutation for a class of DC-DC buck converter systems (BCS). First, a GESO is designed to estimate the total disturbance together with the system state. Then, by choosing an appropriate disturbance-compensation gain, a composite SMC law is designed to attenuate the influence of the parameter uncertainty and reference input mutation on the system output. Both the stability criterion and deign procedure of the system are given. Finally, simulation results show that the designed GESO-based SMC system for the DC-DC BCS is robustly stable and achieves both satisfactory transient and steady-state performance. Comparisons demonstrate that the proposed method provides better transient and steady-state performance for both disturbance rejection and tracking control than either conventional SMC or ESO-based control approach does.
Fast fluorescent blood sugar sensing using phenylboronic acid functionalized N, S-doped carbon dots
Wang Xiaoge,Fan Xiangze,Zhang Bowen,Zhan Mengke,Zhu Jinhua,Hu Weiping,Liu Xiuhua 한국탄소학회 2024 Carbon Letters Vol.34 No.5
A phenylboric acid functionalized carbon dot (2-FPBA-CD) for rapid fluorescent sensing of glucose in blood was synthesized by simply mixing N, S-doped carbon dots (CDs) with phenylboric acid at room temperature. At pH 7.4, the response of 2-FPBA-CD to glucose could reach equilibrium in a very short time (10 min), with a wide responsive linear range of 19.70 µM to 2.54 mM, which can be applied to the detection of glucose in serum. The mechanism studies showed that the layered carbon film of 2-FPBA-CD aggregated after adding glucose, thereby leading to the fluorescence quenching of 2-FPBA-CD.
Discovery of the leinamycin family of natural products by mining actinobacterial genomes
Pan, Guohui,Xu, Zhengren,Guo, Zhikai,Hindra,Ma, Ming,Yang, Dong,Zhou, Hao,Gansemans, Yannick,Zhu, Xiangcheng,Huang, Yong,Zhao, Li-Xing,Jiang, Yi,Cheng, Jinhua,Van Nieuwerburgh, Filip,Suh, Joo-Won,Duan National Academy of Sciences 2017 PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF Vol.114 No.52
<P>Nature's ability to generate diverse natural products from simple building blocks has inspired combinatorial biosynthesis. The knowledge-based approach to combinatorial biosynthesis has allowed the production of designer analogs by rational metabolic pathway engineering. While successful, structural alterations are limited, with designer analogs often produced in compromised titers. The discovery-based approach to combinatorial biosynthesis complements the knowledge-based approach by exploring the vast combinatorial biosynthesis repertoire found in Nature. Here we showcase the discovery-based approach to combinatorial biosynthesis by targeting the domain of unknown function and cysteine lyase domain (DUF-SH) didomain, specific for sulfur incorporation from the leinamycin (LNM) biosynthetic machinery, to discover the LNM family of natural products. By mining bacterial genomes from public databases and the actinomycetes strain collection at The Scripps Research Institute, we discovered 49 potential producers that could be grouped into 18 distinct clades based on phylogenetic analysis of the DUF-SH didomains. Further analysis of the representative genomes from each of the clades identified 28 lnm-type gene clusters. Structural diversities encoded by the LNM-type biosynthetic machineries were predicted based on bioinformatics and confirmed by in vitro characterization of selected adenylation proteins and isolation and structural elucidation of the guangnanmycins and weishanmycins. These findings demonstrate the power of the discovery-based approach to combinatorial biosynthesis for natural product discovery and structural diversity and highlight Nature's rich biosynthetic repertoire. Comparative analysis of the LNM-type biosynthetic machineries provides outstanding opportunities to dissect Nature's biosynthetic strategies and apply these findings to combinatorial biosynthesis for natural product discovery and structural diversity.</P>