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Chang-Liang Xia,Zhe Xu,Jia-Xin Zhao 전력전자학회 2015 JOURNAL OF POWER ELECTRONICS Vol.15 No.1
This paper proposes a novel direct power control (DPC) strategy for neutral-point-clamped (NPC) three-level rectifiers, to directly control the active power, the reactive power and the neutral point potential of the rectifiers by referring to three pre-calculated vector influence tables and minimizing an objective function. In the three vector influence tables, the influences of different voltage vectors on the active power, the reactive power and the neutral-point potential are shown explicitly. A conceptual description and control algorithm of the proposed controller are presented in this paper. Then, numerical simulations and experiments are carried out to validate the proposed method. Both the simulation and experimental results show that good performances during both the steady-state and transient operating conditions are achieved. As a result, the proposed strategy has been proven to be effective for NPC three-level rectifiers.
Xia, Chang-Liang,Xu, Zhe,Zhao, Jia-Xin The Korean Institute of Power Electronics 2015 JOURNAL OF POWER ELECTRONICS Vol.15 No.1
This paper proposes a novel direct power control (DPC) strategy for neutral-point-clamped (NPC) three-level rectifiers, to directly control the active power, the reactive power and the neutral point potential of the rectifiers by referring to three pre-calculated vector influence tables and minimizing an objective function. In the three vector influence tables, the influences of different voltage vectors on the active power, the reactive power and the neutral-point potential are shown explicitly. A conceptual description and control algorithm of the proposed controller are presented in this paper. Then, numerical simulations and experiments are carried out to validate the proposed method. Both the simulation and experimental results show that good performances during both the steady-state and transient operating conditions are achieved. As a result, the proposed strategy has been proven to be effective for NPC three-level rectifiers.
Xia, Shuai,Wang, Xiu-Hua,Liu, Ji-Qiang,Liu, Chang,Chen, Jian-Bin,Zuo, Hua,Xie, Yong-Sheng,Dong, Wen-Liang,Shin, Dong-Soo Korean Chemical Society 2014 Bulletin of the Korean Chemical Society Vol.35 No.6
A facile and effective method has been developed for the synthesis of a novel series of benzofuran derivatives via N-acylation, O-alkylation and intramolecular condensation reactions, starting from readily available substituted o-hydroxy aryl ketone, and chloroacetyl arylamides. This metal-free transition process is characterized by mild reaction conditions, atom economy, short reaction time and a high yield with a decreased amount of by-products.
Shuai Xia,Xiu-Hua Wang,Ji-Qiang Liu,Chang Liu,Jian-Bin Chen,Hua Zuo,Yong-Sheng Xie,Wen-Liang Dong,Dong Soo Shin 대한화학회 2014 Bulletin of the Korean Chemical Society Vol.35 No.6
A facile and effective method has been developed for the synthesis of a novel series of benzofuran derivatives via N-acylation, O-alkylation and intramolecular condensation reactions, starting from readily available substituted o-hydroxy aryl ketone, and chloroacetyl arylamides. This metal-free transition process is characterized by mild reaction conditions, atom economy, short reaction time and a high yield with a decreased amount of by-products.
Fu-Liang Han,Shou-Mei Jiang,Jian-Jun He,Qiu-Hong Pan,Chang-Qing Duan,Ming-Xia Zhang 한국식품과학회 2009 Food Science and Biotechnology Vol.18 No.3
Anthocyanins are considered one of the main color determinants in aged red wine. The anthocyanins in aged red wine made from ‘Cabernet Gernischet’ (Vitis vinifera L. cv.) grape were investigated by high performance liquid chromatography- electronic spray ionization- mass spectrometry (HPLC-ESI-MS) and their color presented in aqueous solution were evaluated using partial least square regression (PLS). The results showed that there were 37 anthocyanins identified in this wine, including 22 pyranoanthocyanins. The analysis of PLS indicated that different anthocyanins showed distinct color values: malvidin 3-O-(6-O-acetyl)-glucoside-4-vinylguaiacol (Mv3-acet-glu-vg) presented the highest color values, while malvidin 3-O-glucoside (Mv3-glu) showed least. Among the free non-acylated anthocyanins, peonidin 3-Oglucoside (Pn3-glu) showed the highest color values; the coumarylated anthocyanins presented higher color values than their corresponding acetylated anthocyanins and parent anthocyanins; pyranoanthocyanins presented also higher color values than their original anthocyanins; the color of anthocyanins depended on their structure. This work will be helpful to reveal evolution in aged red wine.
Jiang, Chang,Liao, Fang-Xin,Rong, Yu-Ming,Yang, Qiong,Yin, Chen-Xi,He, Wen-Zhuo,Cai, Xiu-Yu,Guo, Gui-Fang,Qiu, Hui-Juan,Chen, Xu-Xian,Zhang, Bei,Xia, Liang-Ping Asian Pacific Journal of Cancer Prevention 2014 Asian Pacific journal of cancer prevention Vol.15 No.13
Objective: To compare the efficacy of taxane-based regimens in the first line setting retrospectively in Chinese patients with recurrent and/or metastatic esophageal cancer. Methods: We analyzed 102 recurrent and/or metastatic esophageal cancer patients who received taxanes-based regimens in a first-line setting from January 2009 to December 2013. Sixteen (15.7%) patients were administered Nab-PTX based chemotherapy and 86 patients (84.3%) received paclitaxel (PTX) or docetaxel (DTX) based chemotherapy. Patients in the PTX/DTX group could be further divided into TP (71 patients) and TPF (15 patients) groups. Results: The objective response rate (ORR) of all patients was 20.6%, and the disease control rate (DCR) was 67.6%. The median overall survival (OS) was 10.5 months (95% CI 10.1-16.4) and the median progression-free survival (PFS) was 6.04 months (95% CI 5.09-7.91). The DCR was higher in the TPF group than the TP group (93.3% vs. 59.1%; p = 0.015 ). There were no significant differences in ORR, OS, and PFS among Nab-PTX, TPF and TP groups. Conclusions: The three regimens of Nab-PTX based, TP and TPF proved active in a first line setting of Chinese patients with recurrent and/or metastatic esophageal cancer, and should thus be regarded as alternative treatments.
Once-weekly Subcutaneous Administration of Bortezomib in Patients with Multiple Myeloma
Wang, Liang,Wang, Ke-Feng,Chang, Bo-Yang,Chen, Xiao-Qin,Xia, Zhong-Jun Asian Pacific Journal of Cancer Prevention 2015 Asian Pacific journal of cancer prevention Vol.16 No.5
In patients with multiple myeloma (MM), once-weekly intravenous injection or twice-weekly subcutaneous injection (SC) of bortezomib has been proven to offer non-inferior efficacy to standard twice-weekly intravenous administration, with an improved safety profile. However, whether once-weekly SC bortezomib can further reduce the incidence rate of peripheral neuropathy (PN) and not compromise the efficacy remains to be investigated. 25 patients of MM treated with once-weekly SC bortezomib were reviewed in this study. The median treatment cycles were 4 (range, 2-9 cycles). Complete response (CR) rate was 52%, ${\geq}$very good partial response (VGPR) rate was 72%, and ${\geq}$partial response (PR) rate was 84%. 1-year and 2-year PFS rate was 63.0% and 34.3%, respectively, and 2-year OS rate was 100%. Any grade of PN was reported in 9 patients (36.0%), with 7 patients (28.0%) had grade 1 PN, and 2 patients (8.0%) had grade 2 PN. No patients reported grade 3/4 PN in this cohort. In conclusion, once-weekly subcutaneous administration of bortezomib offers excellent efficacy with a further improved safety profile, especially with regard to PN. It needs to be validated in future prospective randomized trials.
Xiang Zou,Chang-fa Chen,Xia-chang Qi,Jiang-chao Qian,Ju Chu,Ying-ping Zhuang,Si-liang Zhang,Wei Zeng,Wan-jun Li 한국생물공학회 2010 Biotechnology and Bioprocess Engineering Vol.15 No.6
Improvement of Erythromycin A (Er-A) production and purity by metabolic engineering of the industrial erythromycin-producing strains Saccharopolyspora erythraea strians ZL1004 and ZL1007, in which the amounts of tailoring enzymes EryK (a P450 hydroxylase)and EryG (an S-adenosylmethionine-dependent O-methyltransferase)for biotransformation of Erythromycin D to Er-A were modulated, was performed in a 50 L fermentor. Addition of 15 g/L of corn steep liquor to the medium increased Er-A production; maximum Er-A production was 8,196 U/mL at 191 h, which was 81.8% higher than that of control (4,507 U/mL at 184 h). Er-B impurities were completely eliminated, whereas Er-C impurities were only 153 U/mL at 191 h. Analysis of intra- and extracellular metabolites and key enzyme activities in central carbon metabolism revealed that the pool of TCA cycle intermediates was enhanced by the addition of corn steep liquor and induced an increase in erythromycin biosynthesis. There were no significant differences between strains ZL1004 and ZL1007 regarding Er-A production and impurity accumulation. Compared to wild type strain,Er-A production was improved by 23.9% while Er-C was reduced by 83.9% and Er-B was completely eliminated. Furthermore, fermentation of recombinant strain ZL1004was successfully scaled up from laboratory scale (50 L fermentor) to industrial scale (25 and 132 m3), with similar levels of Er-A production and purity obtained.
Wei Li,Chang-Ji Zheng,Liang-Peng Sun,Ming-Xia Song,Yan Wu,Yin-Jing Li,Yi Liu,Hu-Ri Piao 대한약학회 2014 Archives of Pharmacal Research Vol.37 No.7
A series of arylhydrazone derivatives bearing arhodanine moiety have been synthesized, characterized, andevaluated as antibacterial agents. Some of these compoundsshowed potent antibacterial activities against several differentstrains of Gram-positive bacteria, including multidrug-resistant clinical isolates. Of the compounds tested, IIkand IIIk were identified as the most effective, with minimuminhibitory concentration values of 2–4 lg/mL against multidrug-resistant Gram-positive organisms, including methicillin-resistant and quinolone-resistant Staphylococcusaureus. None of the compounds exhibited any activityagainst the Gram-negative bacteria Escherichia coli 1356 at64 lg/mL.